Asbill, C., Kim, N., El-Kattan, A., et al. (2000). Evaluation of a human bio-engineered skin equivalent for drug permeation studies. Pharm. Res. 17, 1092-1097.
Basak, S.C., Mills, D. & Mumtaz, M.M. (2007). A quantitative structure-activity relationship ((Q)SAR) study of dermal absorption using theoretical molecular descriptors. SAR QSAR Environ. Res. 18, 45-55.
Baynes, R.E., Xia, X.R., Imran, M. & Riviere, J.E. (2008). Quantification of Chemical Mixture Interactions Modulating Dermal Absorption Using a Multiple Membrane Fiber Array. Chem. Res. Toxicol. 21, 591-599.
Blackburn, K., Stickney, J.A., Carlson-Lynch, H.L., et al. (2005). Application of the threshold of toxicological concern approach to ingredients in personal and household care products. Regul. Toxicol. Pharmacol. 43, 249-259.
Brain, K.R., Walters, K.A., James, V.J., et al. (1995). Percutaneous penetration of dimethylnitrosamine through human skin in vitro: application from cosmetic vehicles. Food Chem. Toxicol. 33, 315-322.
Brain, K.R., Walters, K.A., Green, D.M., et al. (2005). Percutaneous penetration of diethanolamine through human skin in vitro: application from cosmetic vehicles. Food Chem. Toxicol. 43, 681-690.
Carver, M.P., Williams, P.L. & Riviere, J.E. (1989). The isolated perfused porcine skin flap. III. Percutaneous absorption pharmacokinetics of organophosphates, steroids, benzoic acid, and caffeine. Toxicol. Appl. Pharmacol. 97, 324-337.
Chen, X., Murawski, A., Patel, K., et al. (2008). A Novel Design of Artificial Membrane for Improving the PAMPA Model. Pharm. Res. Jan. 10, 2008. [Epub ahead of print.]
Davies, D.J., Ward, R.J. & Heylings, J.R. (2004). Multi-species assessment of electrical resistance as a skin integrity marker for in vitro percutaneous absorption studies. Toxicol. In Vitro. 18, 351-358.
Diembeck, W., Eskes, C., Heylings, J.R., et al. (2005). Skin absorption and penetration. Altern. Lab Anim. 33, Suppl.1, 105-107.
Dolan, D.G., Naumann, B.D., Sargent, E.V., et al. (2005). Application of the threshold of toxicological concern concept to pharmaceutical manufacturing operations. Regul. Toxicol. Pharmacol. 43, 1-9.
ECVAM. (2002). Biokinetics. Altern. Lab. Anim. 30, Suppl. 1, 56-57.
Fujiwara, S., Yamashita, F. & Hashida, M. (2003). QSAR analysis of interstudy variable skin permeability based on the "latent membrane permeability" concept. J. Pharm. Sci. 92, 1939-1946.
Gamer, A.O., Leibold, E. & van Ravenzwaay, B. (2006). The in vitro absorption of microfine zinc oxide and titanium dioxide through porcine skin. Toxicol. In Vitro. 20, 301-307.
Geinoz, S., Guy, R.H., Testa, B. & Carrupt, P.A. (2004). Quantitative structure-permeation relationships (QSPeRs) to predict skin permeation: a critical evaluation. Pharm. Res. 21, 83-92.
Gibbs, S., van de Sandt, J.J, Merk, H.F, et al. (2007).Xenobiotic metabolism in human skin and 3D human skin reconstructs: a review. Curr. Drug Metab. 8, 758-772.
Katritzky, A.R., Dobchev, D.A., Fara, D.C., et al. (2006). Skin permeation rate as a function of chemical structure. J. Med. Chem. 49, 3305-3314.
Kiss, B., Bíró, T., Czifra, G., et al. (2008). Investigation of micronized titanium dioxide penetration in human skin xenografts and its effect on cellular functions of human skin-derived cells. Exp. Dermatol. Feb. 27, 2008. [Epub ahead of print.]
Kroes, R., Galli, C., Munro, I., et al. (2000). Threshold of toxicological concern for chemical substances present in the diet: a practical tool for assessing the need for toxicity testing. Food Chem. Toxicol. 38, 255-312.
Kroes, R., Renwick, A.G., Cheeseman, M., et al. (2004). Structure-based thresholds of toxicological concern (TTC): guidance for application to substances present at low levels in the diet. Food Chem. Toxicol. 42, 65-83.
Kroes, R., Renwick, A.G., Feron, V., et al. (2007). Application of the threshold of toxicological concern (TTC) to the safety evaluation of cosmetic ingredients. Food Chem. Toxicol. 45, 2533-2562.
Kuntsche, J., Bunjes, H., Fahr, A., et al. (2008). Interaction of lipid nanoparticles with human epidermis and an organotypic cell culture model. Int. J. Pharm. 354, 180-195.
Lian, G., Chen, L. & Han, L. (2008). An evaluation of mathematical models for predicting skin permeability. J. Pharm. Sci. 97, 584-598.
Luo, W., Medrek, S., Misra, J. & Nohynek, G.J. (2007). Predicting human skin absorption of chemicals: development of a novel quantitative structure activity relationship. Toxicol. Ind. Health. 23, 39-45.
Macpherson, S.E., Barton, C.N. & Bronaugh, R.L. (1996). Use of in vitro skin penetration data and a physiologically based model to predict in vivo blood levels of benzoic acid. Toxicol. Appl. Pharmacol. 140, 436-443.
Marjukka Suhonen, T., Pasonen-Seppänen, S., Kirjavainen, M., et al. (2003). Epidermal cell culture model derived from rat keratinocytes with permeability characteristics comparable to human cadaver skin. Eur. J. Pharm. Sci. 20, 107-113.
Mavon, A., Miquel, C., Lejeune, O., et al. (2007). In vitro percutaneous absorption and in vivo stratum corneum distribution of an organic and a mineral sunscreen. Skin Pharmacol. Physiol. 20, 10-20.
Munro, I.C., Ford, R.A., Kennepohl, E. & Sprenger, J.G. (1996). Correlation of structural class with no-observed-effect levels: a proposal for establishing a threshold of concern. Food Chem. Toxicol. 34, 829-867.
Neumann, D., Kohlbacher, O., Merkwirth, C. & Lengauer, T. (2006). A fully computational model for predicting percutaneous drug absorption. J. Chem. Inf. Model. 46, 424-429.
OECD. (2004a). Guidance Document for the Conduct of Skin Absorption Studies. OECD Series on Testing and Assessment. No. 28. OECD. Paris, France. Available here.
OECD. (2004b). Skin absorption: In vivo method. OECD Guidelines for the Testing of Chemicals. Test No. 427. OECD. Paris, France. Available here.
OECD. (2004c). Skin absorption: In vitro method. OECD Guidelines for the Testing of Chemicals. Test No. 428. OECD. Paris, France. Available here.
Ottaviani, G., Martel, S. & Carrupt, P.A. (2006). Parallel artificial membrane permeability assay: a new membrane for the fast prediction of passive human skin permeability. J. Med. Chem. 49, 3948-3954.
Pappinen, S., Tikkinen, S., Pasonen-Seppänen, S., et al. (2007). Rat epidermal keratinocyte organotypic culture (ROC) compared to human cadaver skin: the effect of skin permeation enhancers. Eur. J. Pharm. Sci. 30, 240-250.
Riviere, J.E., Baynes, R.E. & Xia, X.R. (2007). Membrane-coated fiber array approach for predicting skin permeability of chemical mixtures from different vehicles. Toxicol. Sci. 99, 153-161.
Riviere, J.E. & Brooks, J.D. (2007). Prediction of dermal absorption from complex chemical mixtures: incorporation of vehicle effects and interactions into a QSAR framework. SAR QSAR Environ. Res. 18, 31-44.
Schäfer-Korting, M., Bock, U., Gamer, A., et al. (2006). Reconstructed human epidermis for skin absorption testing: results of the German prevalidation study. Altern. Lab. Anim. 34, 283-294.
Schreiber, S., Mahmoud, A., Vuia, A., et al. (2005). Reconstructed epidermis versus human and animal skin in skin absorption studies. Toxicol. In Vitro. 19, 813-822.
Stinchcomb, A.L. (2003). Xenobiotic bioconversion in human epidermis models. Pharm. Res. 20, 1113-1118.
van de Sandt, J.J., van Burgsteden, J.A., Cage, S., et al. (2004). In vitro predictions of skin absorption of caffeine, testosterone, and benzoic acid: a multi-centre comparison study. Regul. Toxicol. Pharmacol. 39, 271-281.
van de Sandt, J.J., Dellarco, M. & Van Hemmen, J.J. (2007). From dermal exposure to internal dose. J. Expo. Sci. Environ. Epidemiol. Suppl. 1, S38-S47.
Van der Merwe, D. & Riviere, J.E. (2005). Comparative studies on the effects of water, ethanol and water/ethanol mixtures on chemical partitioning into porcine stratum corneum and silastic membrane. Toxicol. In Vitro. 19, 69-77.
Van der Merwe, D., Brooks, J.D., Gehring, R., et al. (2006). A physiologically based pharmacokinetic model of organophosphate dermal absorption. Toxicol. Sci. 89, 188-204.
Walters, K.A., Brain, K.R., Dressler, W.E., et al. (1997). Percutaneous penetration of N-nitroso-N-methyldodecylamine through human skin in vitro: application from cosmetic vehicles. Food Chem. Toxicol. 35, 705-712.
Wilkinson, S.C., Maas, W.J., Nielsen, J.B., et al. (2006). Interactions of skin thickness and physicochemical properties of test compounds in percutaneous penetration studies. Int. Arch. Occup. Environ. Health. 79, 405-413.
Xia X.R., Baynes R.E., Monteiro-Riviere, N.A., et al. (2003). A novel in-vitro technique for studying percutaneous permeation with a membrane-coated fiber and gas chromatography/mass spectrometry: part I. Performances of the technique and determination of the permeation rates and partition coefficients of chemical mixtures. Pharm. Res. 20, 275-282.
Xia, X.R., Baynes, R.E., Monteiro-Riviere, N.A. & Riviere, J.E. (2007). An experimentally based approach for predicting skin permeability of chemicals and drugs using a membrane-coated fiber array. Toxicol. Appl. Pharmacol. 221, 320-328.
Zghoul, N., Fuchs, R., Lehr, C.M. & Schaefer, U.F. (2001). Reconstructed skin equivalents for assessing percutaneous drug absorption from pharmaceutical formulations. ALTEX. 18, 103-106.
|
